therapeutic 1,144 words KG: ent-gene-d289a3d6
Contents

nrf2-activators-parkinsons-disease

🔬 Protein Info
Gene Symbolent-gene-d289a3d6
CategoryDisease-Modifying Therapy
TargetNRF2 (NFE2L2) / KEAP1 Pathway
Development StagePhase I-II
Route of AdministrationOral
Key CompoundsSulforaphane, Dimethyl fumarate, Bardoxolone methyl
ModelFinding
MPTP model40-60% dopaminergic neuron protection
6-OHDA model35-45% neurodegeneration attenuation
Alpha-synuclein overexpressionEnhanced autophagic clearance of α-synuclein
Drosophila PD modelExtended lifespan, preserved climbing ability
PopulationDose
Early PD100-200 μmol/day (~17-35 mg SFN)
Prodromal40-100 μmol/day
TrialPhase
NCT04550494Phase II
KG Connections2 knowledge graph edges
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (3)

Epigenetic Memory Reprogramming via CRISPRa-Mediated Chromat
Score: 0.52
Matrix Stiffness Normalization via Targeted Lysyl Oxidase In
Score: 0.51
Sphingomyelin Synthase Activators for Raft Remodeling
Score: 0.47

Related Analyses (16)

Lipid raft composition changes in synaptic neurodegeneration
neurodegeneration · completed
TREM2 agonism vs antagonism in DAM microglia
neurodegeneration · failed
TDP-43 phase separation therapeutics for ALS-FTD
neurodegeneration · archived
Blood-brain barrier transport mechanisms for antibody therap
neurodegeneration · archived
What are the mechanisms by which gut microbiome dysbiosis in
neurodegeneration · completed

Related Experiments (4)

Acteoside treatment in LPS-induced SALI mouse model
validation · proposed · Score: 0.90
Nrf2 inhibitor ML385 mechanism validation experiment
exploratory · proposed · Score: 0.85
Acteoside effects on RAW264.7 macrophage cells
exploratory · proposed · Score: 0.85
Cytochrome Therapeutics
clinical · proposed · Score: 0.40

Knowledge Graph (2 edges)

ent-gene-d289a3d6 data_in benchmark_ot_ad_answer_key:NRF2
benchmark_ot_ad_answer_key:NRF2 data_in ent-gene-d289a3d6