S-equol-induced ferroptosis mechanism in TNBC cells

Exploratory Score: 0.900 Price: $0.50 Triple negative breast cancer TNBC cell lines Status: proposed

What This Experiment Tests

Exploratory experiment designed to discover new patterns targeting PPARγ, GPX4, NCOA4 in TNBC cell lines. Primary outcome: Ferroptosis induction markers (lipid peroxidation, Fe²+ levels)

Description

Mechanistic studies investigating how S-equol induces ferroptosis in triple negative breast cancer cells through modulation of the PI3K/AKT/mTOR signaling pathway. The experiments examined the effects of S-equol on lipid peroxidation levels, intracellular Fe²+ concentrations, and key ferroptosis regulators including PPARγ, GPX4, and NCOA4. The study utilized specific agonists for PPARγ and STAT3, as well as autophagy inhibitor ULK101, to validate the proposed mechanism. Additionally, NCOA4 knockdown and PPARγ overexpression experiments were performed to further confirm the molecular pathways involved in S-equol-mediated ferroptosis induction.

TARGET GENE
PPARγ, GPX4, NCOA4
MODEL SYSTEM
TNBC cell lines
ESTIMATED COST
$0
TIMELINE
0 months
PATHWAY
PI3K/AKT/mTOR signaling pathway, ferroptosis, ferritinophagy
SOURCE
extracted_from_pmid_41925800
PRIMARY OUTCOME
Ferroptosis induction markers (lipid peroxidation, Fe²+ levels)

Scoring Dimensions

Info Gain 0.00 (25%) Feasibility 0.00 (20%) Hyp Coverage 0.00 (20%) Cost Effect. 0.00 (15%) Novelty 0.00 (10%) Ethical Safety 0.00 (10%) 0.900 composite

📖 Wiki Pages

GPX4 Protein - Glutathione Peroxidase 4proteinGPX4 (Glutathione Peroxidase 4)proteinSTAT3 ProteinproteinPI3K p110α ProteinproteinPI3K ProteinproteinNCOA4 ProteinproteinGPX4** is a protein. This page describes its strucredirectakt-proteinproteinpi3k-akt-signalingmechanismPI3K/Akt Signaling in Parkinson's DiseasemechanismPI3K-Akt Signaling in Parkinson's DiseasemechanismPI3K/Akt Signaling in NeurodegenerationmechanismPI3K/AKT/mTOR Signaling Pathway in NeurodegeneratimechanismSTAT3 GenegenePI3K — Phosphoinositide 3-Kinasegene

Protocol

Lipid peroxidation assays, iron level measurement, gene knockdown/overexpression, pharmacological inhibition

Expected Outcomes

Increased lipid peroxidation and Fe²+ levels, decreased GPX4 activity

Success Criteria

Significant changes in ferroptosis markers upon S-equol treatment

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