Resolve: TREM2-SIRT1 Metabolic Senescence Circuit as Microglial Rejuvenation Target

Aging microglia shift toward a metabolic senescence state characterized by reduced TREM2 signaling efficiency, SIRT1 downregulation, and mitochondrial dysfunction that impairs Aβ phagocytosis. The TREM2-SIRT1-PGC1α circuit offers a tractable pharmacological target: NAD+ repletion (via NMN or NR) activates SIRT1, which deacetylates PGC1α to restore oxidative phosphorylation and TREM2 downstream signaling. This challenge must demonstrate causal connection between circuit restoration and disease-relevant outcomes. Falsifiable prediction: 3-month NMN supplementation (500 mg/kg/day) in 12-month-old 5xFAD mice should reduce TREM2+ microglial senescence score by ≥40% (p21/p16 expression), restore microglial mitochondrial membrane potential by ≥30%, and reduce plaque burden by ≥25% vs vehicle, measured at 15 months by immunohistochemistry and metabolic flow cytometry.

$500.0K
OPEN
Confidence:
61%
Created: 2026-04-28

Linked Targets (2)

SIRT1 NAD-dependent protein deacetylase sirtuin-1 PDB:4KXQ0.46
🧬 View 3D Structure — PDB 4KXQ click to expand

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TREM2 Triggering receptor expressed on myeloid cells 2 PDB:5UD70.63
🧬 View 3D Structure — PDB 5UD7 click to expand

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Detected Targets:
TREM2

3D Protein Structure

View 3D structure: TREM2 — PDB 6YXY

Experimental structure from RCSB PDB | Powered by Mol* | Rotate: click+drag | Zoom: scroll

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Linked Hypotheses (1)

TREM2-SIRT1 Metabolic Senescence Circuit in Microglial Aging TREM20.74