| Gene Symbol | 5-HT2A RECEPTOR |
| Aliases | HTR2A |
| Chromosome | 13q14 |
| Molecular Weight | 53 kDa |
| Strategy | Mechanism |
| 5-HT2A Antagonists (nelotanserin) | Reduce LID |
| 5-HT2A Inverse Agonists | Stabilize inactive state |
| Allosteric Modulators | Enhance therapeutic signaling |
| Compound | Selectivity |
| Psilocybin | 5-HT2A agonist |
| LSD | 5-HT2A/5-HT1A agonist |
| DMT | 5-HT2A agonist |
| Clozapine | 5-HT2A/D2 antagonist |
| Risperidone | 5-HT2A/D2 antagonist |
| Nelotanserin | 5-HT2A inverse agonist |
| Databases | GeneCardsUniProtNCBI GeneHPASTRING |