therapeutic 1,745 words KG: ent-gene-45b60f3e 2026-03-22
kind:therapeuticsection:therapeuticsstate:published
Contents

COMT Inhibitors

🔬 Protein Info
Gene Symbolent-gene-45b60f3e
FeatureEntacapone
GenerationFirst
DosingWith each levodopa dose
COMT inhibition~65%
CNS penetrationNo
ON time increase1-2 hours
Hepatotoxicity riskNo
Liver monitoringNot required
Approval year1998/1999
DrugSelectivity
EntacaponeSelective
TolcaponeNon-selective
OpicaponeSelective
ParameterWith COMT-I
OFF time reduction1-2 hours
KG Connections2 knowledge graph edges
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

Knowledge Graph