mechanism 1,855 words KG: ent-gene-694200ea 2026-04-02
kind:mechanismsection:mechanismsstate:publishedevidence:strong
Contents

GBA and Lysosomal Function in Parkinson's Disease

🔬 Protein Info
Gene Symbolent-gene-694200ea
Loss-of-function (LoF) allelesN370S, L444P, 84insGG, Rec1 (del55), and many others.
Missense mutationsE326K, T369M, which are common in European populations.
Complex allelesrecombinant alleles that can have variable enzymatic activity.
ReactionGlcCer + H2O → Ceramide + Glucose.
LocationLysosomal lumen, mediated by the integral membrane protein GCase, which requires the co-factor **saposin C** for optimal activity.
Saposin Cco-factor; deficiency leads to a variant of GD.
LIMP-2 (SCARB2)transports GCase from the ER to the lysosome.
GCase substrate GlcCeraccumulation impairs lysosomal membrane integrity and can cause **ER stress**[@mazzulli2011].
Cathepsin D (CTSD)the principal protease for alpha-synuclein degradation – shows reduced activity in GBA-deficient neurons.
MacroautophagyImpaired flux prevents efficient clearance of alpha-synuclein aggregates.
Chaperone-mediated autophagy (CMA)GCase deficiency down-regulates LAMP-2A, reducing CMA activity[@avenali2020].
Proteasomal degradationCeramide accumulation can inhibit the 26S proteasome, contributing to a "double-hit" on protein clearance.
Kinase activity cross-regulationGCase deficiency leads to accumulation of glucosylceramide, which directly activates LRRK2 kinase activity through lipid raft reorganization and Rab phosphorylation cascades.
Lysosomal trafficking impairmentLRRK2-mediated phosphorylation of Rab7 and Rab10 disrupts lysosomal trafficking in GBA-deficient neurons, creating a "double-hit" on autophagy[@liu2021].
Synergistic effects on alpha-synucleinCombined GBA loss and LRRK2 hyperactivity dramatically accelerates alpha-synuclein aggregation.
KG Connections2 knowledge graph edges
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (20)

Purinergic Signaling Polarization Control
Score: 0.55
Mechanosensitive Ion Channel Reprogramming
Score: 0.51
Lipid Droplet Dynamics as Phenotype Switches
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Smartphone-Detected Motor Variability Correction
Score: 0.56
Microbial Metabolite-Mediated α-Synuclein Disaggregation
Score: 0.45

Related Analyses (30)

Does TFEB activation directly restore mutant GBA enzyme acti
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GBA-Synuclein Loop: Therapeutic Strategies for Parkinson's D
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Astrocyte reactivity subtypes in neurodegeneration
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Autophagy-lysosome pathway convergence across neurodegenerat
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Related Experiments (30)

Validate Mitochondria-Lysosome Contact Site Dysfunction in P
validation · proposed · Score: 0.40
Alpha-Synuclein Aggregation Triggers — Sporadic PD Initiatio
clinical · proposed · Score: 0.40
Autophagy Enhancement Drug Screening for Neurodegeneration
clinical · proposed · Score: 0.40
Genetic Risk Modifiers in DLB Phenotype
clinical · proposed · Score: 0.40
DLB Treatment Response Biomarkers — Predicting Cholinesteras
clinical · proposed · Score: 0.40

See Also (15)

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Knowledge Graph (2 edges)

ent-gene-694200ea data_in benchmark_ot_ad_answer_key:GBA
benchmark_ot_ad_answer_key:GBA data_in ent-gene-694200ea