idea 616 words KG: ent-gene-8c4b5215 2026-03-21
kind:ideakind:therapy-ideasection:ideasstate:published
Contents

GFAP-Guided Astrocyte Modulation Therapy

🔬 Protein Info
Gene SymbolGFAP
Full NameGuided Astrocyte Modulation Therapy
AliasesGlial Fibrillary Acidic Protein Gene, Glial Fibrillary Acidic Protein
Chromosome17q21.31
Protein FamilyType III intermediate filament protein
Protein TypeBiomarker / Structural Protein
Target ClassStructural Protein
FunctionBiomarker readout — GFAP levels reflect astrocyte reactivity; modulating upstream pathways (e.g., NF-κB, JAK-STAT) reduces GFAP expression
Mechanism of ActionBiomarker readout — GFAP levels reflect astrocyte reactivity; modulating upstream pathways (e.g., NF-κB, JAK-STAT) reduces GFAP expression
Primary ExpressionCytoplasm (cytoskeletal intermediate filament)
DruggabilityMedium (0.52)
Clinical StagePhase II
Molecular Weight50 kDa
Amino Acids432 aa
Exons9
PathwaysAmyloid, Er Stress, Inflammasome, Innate Immunity, Mapk
UniProt IDP14136
GeneCardsGFAP
Human Protein AtlasGFAP
Associated DiseasesALEXANDER_DISEASE, ALS, ALZHEIMER'S DISEASE, ALZHEIMER_DISEASE, ASTROGLIAL_ACTIVATION, AXONAL DEGENERATION
Known Drugs/CompoundsMETFORMIN, VANADIUM, TMT, PHENYTOIN, DSS, Hormones
InteractionsMMP9, TNF, TLR4, MMP2, TMEM119, NFL
SciDEX TargetView Target Profile (8 clinical trials)
SciDEX HypothesesHeterogeneous astrocyte activation states differen
GFAP-Positive Reactive Astrocyte Subtype Delineati
KG Connections3103 knowledge graph edges
DatabasesGeneCardsNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (30)

Bacterial Enzyme-Mediated Dopamine Precursor Synthesis
Score: 0.36
Heterogeneous astrocyte activation states differentially imp
Score: 0.52
Astrocyte-Mediated Microglial Memory Erasure
Score: 0.46
GFAP-Positive Reactive Astrocyte Subtype Delineation
Score: 0.52
Gamma entrainment therapy to restore hippocampal-cortical sy
Score: 0.68

Related Analyses (30)

Neuroinflammation and microglial priming in early Alzheimer'
neurodegeneration · archived
Mechanistic validation of SEA-AD differential expression hyp
neurodegeneration · failed
Do these mechanistic hypotheses explain layer-specific synap
neurodegeneration · failed
Do these mechanistic hypotheses from the SEA-AD Atlas bundle
neurodegeneration · failed
TDP-43 phase separation therapeutics for ALS-FTD
neurodegeneration · archived

Related Experiments (30)

iPSC-NPC effects on astrocytes in vitro ICH model
exploratory · proposed · Score: 0.90
Plasma ATN biomarkers across AD continuum in Chilean cohort
clinical · proposed · Score: 0.95
Real-world safety study of Lecanemab in Japanese AD patients
clinical · proposed · Score: 0.95
GWAS of plasma GFAP in East Asian cohort
exploratory · proposed · Score: 0.95
GWAS of composite biomarker score
exploratory · proposed · Score: 0.90

Knowledge Graph (2 edges)

ent-gene-8c4b5215 data_in benchmark_ot_ad_answer_key:GFAP
benchmark_ot_ad_answer_key:GFAP data_in ent-gene-8c4b5215