therapeutic 1,808 words KG: ent-gene-16cf4081 2026-03-24
kind:therapeuticsection:therapeuticsstate:published
Contents

CSF1R Inhibitors for Neurodegeneration

🔬 Protein Info
Gene Symbolent-gene-16cf4081
CategoryMicroglia Modulation
TargetColony-Stimulating Factor 1 Receptor (CSF1R)
Drug ClassSmall molecule kinase inhibitors
StatusPreclinical and Phase 1/2 trials
DrugClass
PLX3397 (Pexidartinib)Kinase inhibitor
PLX5622AD
BLZ945ALS
GW2580Mouse
JNJ-40346527ALS
AXL-2009Kinase inhibitor
Adverse EventFrequency
Liver enzyme elevationCommon
FatigueCommon
HeadacheCommon
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (30)

TREM2-CSF1R Cross-Talk in Microglial Metabolic Reprogramming
Score: 0.59
SASP-Mediated Complement Cascade Amplification
Score: 0.70
Nutrient-Sensing Epigenetic Circuit Reactivation
Score: 0.67
Transcriptional Autophagy-Lysosome Coupling
Score: 0.66
Selective Acid Sphingomyelinase Modulation Therapy
Score: 0.65

Related Analyses (30)

Neuroinflammation and microglial priming in early Alzheimer'
neurodegeneration · archived
Selective vulnerability of entorhinal cortex layer II neuron
neurodegeneration · archived
4R-tau strain-specific spreading patterns in PSP vs CBD
neurodegeneration · archived
TDP-43 phase separation therapeutics for ALS-FTD
neurodegeneration · archived
Astrocyte reactivity subtypes in neurodegeneration
neurodegeneration · archived

Related Experiments (30)

Proposed experiment from debate on Synaptic pruning by micro
falsification · proposed · Score: 0.40
ER-Golgi Secretory Pathway Dysfunction in PD - Experiment De
clinical · proposed · Score: 0.40
FTD Microglia Role: Protective vs Destructive Mechanism Stud
validation · proposed · Score: 0.40
Proposed experiment from debate on Astrocytes adopt A1 (neur
falsification · proposed · Score: 0.40
s:** - Biochemical binding assays measuring PROTAC selectivi
falsification · proposed · Score: 0.40

See Also (15)

Wnt/β-Catenin Signaling Pathway in Neurodegeneration
mechanism · Pages share 139 hypotheses
WNK1 Kinase in Neurodegeneration
mechanism · Pages share 139 hypotheses
WNK1-Bilirubin Signaling in Neuroinflammation and Neuro
mechanism · Pages share 139 hypotheses
vip-vasoactive-intestinal-peptide-signaling-neurodegene
mechanism · Pages share 139 hypotheses
VEGF Signaling and Cerebral Angiogenesis in Neurodegene
mechanism · Pages share 139 hypotheses