entity 1,485 words KG: dopamine 2026-03-23
kind:entitysection:entitiesstate:published
Contents

Dopamine

🔬 Protein Info
Gene Symboldopamine
FunctionInhibits prolactin secretion
Monoamine oxidase (MAO-A and MAO-B)Located on the outer mitochondrial membrane; converts dopamine to 3,4-dihydroxyphenylacetaldehyde (DOPAL), a highly reactive and toxic intermediate
Catechol-O-methyltransferase (COMT)Converts dopamine to 3-methoxytyramine (3-MT)
D1 receptorMost abundant dopamine receptor in the brain; high expression in striatum, cortex, and limbic system. Activates adenylyl cyclase and increases cAMP.
D5 receptorLower expression; found in hippocampus, thalamus, and cortex.
D2 receptorHigh expression in striatum, SNpc, and VTA. Exists in two splice variants: D2S (short, presynaptic autoreceptor) and D2L (long, postsynaptic). Inhibits adenylyl cyclase and decreases cAMP.
D3 receptorExpressed in limbic regions, nucleus-accumbens, and VTA.
D4 receptorLower expression; enriched in frontal cortex and limbic areas.
OriginHypothalamic arcuate nucleus → **Target**: Pituitary gland
Disease relevanceDisruption by dopamine antagonists causes hyperprolactinemia
Associated DiseasesParkinson's Disease
Known Drugs/Compoundsdiabetic retinal neurodegeneration, NRF2, lipopolysaccharide, Ginsenoside Rb1
KG Connections22 knowledge graph edges
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (30)

Circadian Glymphatic Entrainment via Targeted Orexin Recepto
Score: 0.62
Astrocyte-Intrinsic NLRP3 Inflammasome Activation by Alpha-S
Score: 0.60
Microbial Inflammasome Priming Prevention
Score: 0.58
AMPK hypersensitivity in astrocytes creates enhanced mitocho
Score: 0.57
Synthetic Biology BBB Endothelial Cell Reprogramming
Score: 0.57

Related Analyses (30)

4R-tau strain-specific spreading patterns in PSP vs CBD
neurodegeneration · archived
TDP-43 phase separation therapeutics for ALS-FTD
neurodegeneration · archived
Astrocyte reactivity subtypes in neurodegeneration
neurodegeneration · archived
Blood-brain barrier transport mechanisms for antibody therap
neurodegeneration · archived
Microglia-astrocyte crosstalk amplification loops in neurode
neurodegeneration · archived

Related Experiments (30)

iPSC-derived astrocyte-neuron co-culture mitochondrial trans
exploratory · proposed · Score: 0.90
s:** - Dose-response studies showing therapeutic window with
falsification · proposed · Score: 0.40
AAV Serotype Comparison for LRRK2 Knockdown in PD Gene Thera
validation · proposed · Score: 0.40
AAV-LRRK2 IND-Enabling Study Design
clinical · proposed · Score: 0.40
AAV Serotype Comparison for LRRK2 Knockdown in PD
validation · proposed · Score: 0.40

See Also (3)

Alzheimer Indonesia
institution · KG edge: activates
Amyloid-Related Imaging Abnormalities (ARIA)
entity · KG edge: activates
acetylcholine
general · KG edge: co_discussed

Knowledge Graph (12 edges)

dopamine regulates neuronal uptake
dopamine treats diabetic retinal neurodegeneration
dopamine activates NRF2
dopamine regulates GPX4
dopamine regulates BDNF
dopamine expressed_in striatum
dopamine expressed_in mesolimbic circuit
dopamine loss_affects neuron
dopamine loss_affects SNCA
dopamine loss_affects Alzheimer