idea 1,576 words KG: ent-gene-95250f02 2026-03-24
kind:ideakind:therapy-ideasection:ideasstate:published
Contents

cGAS-STING Pathway Inhibition for Chronic Neuroinflammation

🔬 Protein Info
Gene Symbolent-gene-95250f02
Primary ExpressioncGAS and STING are expressed in microglia, astrocytes, and at lower levels in neurons; upregulated in disease states
Subcellular LocalizationcGAS is cytoplasmic (senses dsDNA); STING resides at the ER membrane and traffics to Golgi upon activation
Primary TargetSTING (TMEM173) palmitoylation site or trafficking domain; or cGAS catalytic domain
Target TypeSmall-molecule STING inhibitor (H-151 class) or cGAS inhibitor (RU.521 class)
KG Connections2 knowledge graph edges
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (29)

Bacterial Enzyme-Mediated Dopamine Precursor Synthesis
Score: 0.36
Senescent Cell Mitochondrial DNA Release
Score: 0.54
cGAS-STING Senescence Circuit Disruption
Score: 0.49
White Matter Oligodendrocyte Protection via CXCL10 Inhibitio
Score: 0.48
White Matter Vulnerability Prevention via Oligodendrocyte Pr
Score: 0.47

Related Analyses (19)

What determines the specificity of TDP-43-induced mitochondr
neurodegeneration · failed
How does chronic cGAS/STING activation downstream of TDP-43
neuroinflammation · failed
What upstream mechanisms cause TDP-43 to trigger mPTP openin
neurodegeneration · failed
TDP-43 phase separation therapeutics for ALS-FTD
neurodegeneration · archived
Astrocyte reactivity subtypes in neurodegeneration
neurodegeneration · archived

Related Experiments (18)

Sporadic ALS Initiation Biology: Deep Phenotyping of At-Risk
clinical · proposed · Score: 0.40
cGAS-STING Pathway Validation Study in Parkinson's Disease
clinical · proposed · Score: 0.40
Macroautophagy Dysfunction in PD - Experiment Design
clinical · proposed · Score: 0.40
s:** - Compare brain penetration in FcRn+/+ vs FcRn-/- mice
falsification · proposed · Score: 0.40
s:** - GPR32 knockout in microglia should worsen neuroinflam
falsification · proposed · Score: 0.40

Knowledge Graph (2 edges)

ent-gene-95250f02 data_in benchmark_ot_ad_answer_key:CGAS
benchmark_ot_ad_answer_key:CGAS data_in ent-gene-95250f02