idea 2,450 words KG: ent-gene-3d51813d 2026-03-24
kind:ideakind:therapy-ideasection:ideasstate:published
Contents

GPNMB Modulation for Lipid-Laden Microglia Rescue

🔬 Protein Info
Gene Symbolent-gene-3d51813d
Primary ExpressionLow in homeostatic microglia; massively upregulated (10-50x) in DAM/lipid-laden microglia in AD, PD, GBA-PD, and Gaucher disease[@kerenshaul2017]
Subcellular LocalizationCell surface of activated/dysfunctional microglia; shed ectodomain detectable in CSF
Primary TargetGPNMB (extracellular domain) on lipid-laden microglia
Target TypeAntibody-drug conjugate (ADC) for LLM depletion, or anti-GPNMB agonist antibody to restore phagocytic function
KG Connections2 knowledge graph edges
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (30)

TREM2-Dependent Astrocyte-Microglia Cross-talk in Neurodegen
Score: 0.64
TREM2-Mediated Astrocyte-Microglia Cross-Talk in Neurodegene
Score: 0.61
TREM2-mediated microglial tau clearance enhancement
Score: 0.49
TREM2 Conformational Stabilizers for Synaptic Discrimination
Score: 0.41
Prime Editing Precision Correction of APOE4 to APOE3 in Micr
Score: 0.62

Related Analyses (30)

TDP-43 phase separation therapeutics for ALS-FTD
neurodegeneration · archived
Astrocyte reactivity subtypes in neurodegeneration
neurodegeneration · archived
Blood-brain barrier transport mechanisms for antibody therap
neurodegeneration · archived
Microglia-astrocyte crosstalk amplification loops in neurode
neurodegeneration · archived
APOE4 structural biology and therapeutic targeting strategie
neurodegeneration · archived

Related Experiments (24)

Animal Model Comparison for Neurodegenerative Disease Therap
clinical · proposed · Score: 0.40
Endocannabinoid System Dysfunction Validation in Parkinson's
clinical · proposed · Score: 0.40
Glymphatic-Circadian Axis Enhancement Therapy for Parkinson'
clinical · proposed · Score: 0.40
Gut Microbiome-Derived Metabolites in Alpha-Synuclein Propag
clinical · proposed · Score: 0.40
Neural Oscillation Dysfunction Validation in Parkinson's Dis
clinical · proposed · Score: 0.40

Knowledge Graph (2 edges)

ent-gene-3d51813d data_in benchmark_ot_ad_answer_key:GPNMB
benchmark_ot_ad_answer_key:GPNMB data_in ent-gene-3d51813d