disease 1,147 words KG: ent-dise-1d66a04d 2026-03-21
kind:diseasesection:diseasesstate:published
Contents

APOE4 (Apolipoprotein E4)

Disease Info
InheritanceCo-dominant (alongside APOE2 or APOE3)
GeneAPOE (Apolipoprotein E)
Chromosome19q13.32
SNP IDrs429358 (Arg130), rs7412 (Cys176)
Allele Frequency~15-20% in Caucasian populations; ~10-15% globally
Nucleotide ChangesC at rs429358 (Arg130), T at rs7412 (Cys176)
Increased lipid binding capacityhighest among all APOE isoforms
Domain interactionN-terminal and C-terminal domains interact abnormally
Fragmentation susceptibilityprone to proteolytic cleavage generating neurotoxic fragments
Heterozygotes (E3/E4)3-4x increased risk compared to E3/E3
Homozygotes (E4/E4)10-15x increased risk, with earlier onset (~65-70 years)
Population Attributable Risk~20-25% of AD cases attributable to APOE4 [3]
DatabasesOMIMOrphanetClinicalTrialsPubMed

Knowledge Graph

Related Hypotheses (18)

APOE Isoform Expression Across Glial Subtypes
Score: 0.48
Astrocyte-Selective APOE4 Silencing via Lipid Nanoparticles
Score: 0.53
Selective APOE4 Degradation via Proteolysis Targeting Chimer
Score: 0.59
Synthetic Biology BBB Endothelial Cell Reprogramming
Score: 0.57
Competitive APOE4 Domain Stabilization Peptides
Score: 0.56

Related Analyses (21)

APOE4-driven lipid metabolism dysregulation in astrocytes an
neuroscience · failed
Neuroinflammation and microglial priming in early Alzheimer'
neurodegeneration · archived
Neuroinflammation and microglial priming in early AD
neurodegeneration · completed
Do APOE4-driven senescent astrocytes cause neurodegeneration
neurodegeneration · failed
How does APOE4 mechanistically increase TDP-43 pathology fre
neurodegeneration · failed

Related Experiments (21)

Multi-omics analysis of myricanol effects on gene expression
exploratory · proposed · Score: 0.88
APOE4 association with TDP-43 pathology in AD
exploratory · proposed · Score: 0.75
s:** - Biochemical binding assays measuring PROTAC selectivi
falsification · proposed · Score: 0.40
s:** - Dose-response studies showing therapeutic window with
falsification · proposed · Score: 0.40
AD Amyloid-Resilient Phenotype Study — Why Some amyloid-Posi
clinical · proposed · Score: 0.40

See Also (15)

LRP1-Targeted ApoE-Mimetic Peptide Delivery
idea · Pages share 10 hypotheses
APOE contributes to Alzheimer's disease by regulating b
hypothesis · Pages share 10 hypotheses
LX1001 Phase 1/2 Trial (NCT03634007) - Gene Therapy for
clinical · Pages share 10 hypotheses
vitamin-d-therapy-neurodegeneration
therapeutic · Pages share 9 hypotheses
TREM2 Agonist Therapy for Neurodegeneration
therapeutic · Pages share 9 hypotheses