gene 1,290 words KG: GRK2 2026-03-27
kind:genesection:genesstate:published
Contents

GRK2 — G Protein-Coupled Receptor Kinase 2

🧬 Gene Info
Gene SymbolGRK2
Full NameG Protein-Coupled Receptor Kinase 2
AliasesGRK2/Beta-ARK1
Chromosome11q13.4
Protein FamilyGRK family (PKA/PKG/PKC-like)
Protein TypeKinase
FunctionReceptor Activation — Upon ligand binding, GPCRs undergo conformational changes that enable interaction with heterotrimeric G proteins.
Molecular Weight80 kDa
Amino Acids729 aa
Pathwaysautophagy pathway, complement cascade, phagocytosis
UniProt ID[P10147](https://www.uniprot.org/uniprot/P10147)
Ensembl IDENSG00000188020
OMIM109635
GeneCardsGRK2
Human Protein AtlasGRK2
Associated Diseasesneurodegeneration
Known Drugs/Compoundsrapamycin
InteractionsFOXO1, NR1H3, MAP3K5, SREBF2, NFE2L2, C1Q
KG Connections167 knowledge graph edges
DatabasesGeneCardsNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (11)

Nutrient-Sensing Epigenetic Circuit Reactivation
Score: 0.67
Transcriptional Autophagy-Lysosome Coupling
Score: 0.66
Circadian Glymphatic Entrainment via Targeted Orexin Recepto
Score: 0.62
Smartphone-Detected Motor Variability Correction
Score: 0.56
Heat Shock Protein 70 Disaggregase Amplification
Score: 0.51

Related Analyses (10)

Blood-brain barrier transport mechanisms for antibody therap
neurodegeneration · archived
Microglia-astrocyte crosstalk amplification loops in neurode
neurodegeneration · archived
Perivascular spaces and glymphatic clearance failure in AD
neurodegeneration · archived
Cell type vulnerability in Alzheimers Disease (SEA-AD transc
neurodegeneration · archived
Protein aggregation cross-seeding across neurodegenerative d
neurodegeneration · archived

See Also (6)

CREB-independent Neuronal Survival Pathways
mechanism · KG edge: activates
FOXO1 Gene
gene · KG edge: activates
C1QA Gene — Complement Component 1q A Chain
gene · KG edge: interacts_with
BECN1 Gene
gene · KG edge: interacts_with
Autophagy Enhancement Drug Screening for Neurodegenerat
experiment · KG edge: interacts_with

Knowledge Graph (12 edges)

GRK2 activates HTRA2
GRK2 activates KDM6B
GRK2 activates LAMP2
GRK2 activates LC3
GRK2 activates MAP3K5
GRK2 activates MTOR
GRK2 activates NFE2L2
GRK2 activates NOS3
GRK2 activates NR1H3
GRK2 activates P62