gene 2,267 words KG: apoe
Contents

APOE — Apolipoprotein E

🧬 Gene Info
Gene SymbolAPOE
Full NameApolipoprotein E
Chromosome19q13.32
Target ClassLigand
FunctionIt binds to the LDL receptor family to facilitate uptake of lipoprotein particles.
Mechanism of ActionProtein-protein interaction modulator or lipid metabolism enhancer
DruggabilityMedium (0.47)
Clinical StagePhase II
Molecular Weight34 kDa
PathwaysAmyloid, Autophagy, Blood-Brain Barrier, Brain Lipid Metabolism, Cholesterol
GeneCardsAPOE
Human Protein AtlasAPOE
GenotypeAD Risk
ε3/ε3Baseline (1x)
ε3/ε4~3x increased
Associated DiseasesAD, AGING, ALS, ALZHEIMER, ALZHEIMER'S DISEASE, AMI
Known Drugs/CompoundsLIPOPROTEINS, Triacylglycerol, Lipid-Targeting Therapeutic Strategies
InteractionsLRP1, LDLR, LOX, IL6, SREBF1, PSEN2
SciDEX TargetView Target Profile (8 clinical trials)
SciDEX HypothesesAPOE4-Specific Lipidation Enhancement Therapy
Prime Editing Precision Correction of APOE4 to APO
Selective APOE4 Degradation via Proteolysis Target (+11 more)
KG Connections4776 knowledge graph edges
DatabasesGeneCardsUniProtNCBI GeneHPASTRING

Knowledge Graph

Related Hypotheses (30)

Selective APOE4 Degradation via Proteolysis Targeting Chimer
Score: 0.59
Competitive APOE4 Domain Stabilization Peptides
Score: 0.56
APOE4 Allosteric Rescue via Small Molecule Chaperones
Score: 0.54
Targeted APOE4-to-APOE3 Base Editing Therapy
Score: 0.53
Engineered Apolipoprotein E4-Neutralizing Shuttle Peptides
Score: 0.51

Related Analyses (30)

Lipid metabolism dysregulation and membrane integrity in Alz
neurodegeneration · completed
APOE4 structural biology and therapeutic targeting strategie
neurodegeneration · archived
Mechanistic role of APOE in neurodegeneration
neurodegeneration · archived
CRISPR-based therapeutic approaches for neurodegenerative di
neurodegeneration · archived
Cell type vulnerability in Alzheimers Disease (SEA-AD transc
neurodegeneration · archived

Related Experiments (30)

GWAS of plasma NfL in East Asian cohort
exploratory · proposed · Score: 0.95
GWAS of plasma pTau217 in East Asian cohort
exploratory · proposed · Score: 0.95
Dairy intake and dementia risk in Malmö Diet and Cancer coho
clinical · proposed · Score: 0.95
GWAS of plasma pTau181 in East Asian cohort
exploratory · proposed · Score: 0.95
GWAS of plasma GFAP in East Asian cohort
exploratory · proposed · Score: 0.95

See Also (15)

UPenn Observational Research Repository (NCT04715399)
clinical · Pages share 9 hypotheses
remternetug-anti-amyloid-alzheimers
clinical_trial · Pages share 9 hypotheses
nct05508789
clinical_trial · Pages share 9 hypotheses
LX1001 Long-Term Follow-up (NCT05400330) - Gene Therapy
clinical · Pages share 9 hypotheses
LX1001 Phase 1/2 Trial (NCT03634007) - Gene Therapy for
clinical · Pages share 9 hypotheses

Knowledge Graph (5 edges)

apoe implicated_in neurodegeneration
apoe data_in ad_genetic_risk_loci:APOE
apoe data_in benchmark_ot_ad_answer_key:APOE
ad_genetic_risk_loci:APOE data_in apoe
benchmark_ot_ad_answer_key:APOE data_in apoe