protein 903 words KG: P2RY12PROTEIN 2026-03-21
kind:proteinsection:proteinsstate:published
Contents

P2Y12 Receptor Protein

🔬 Protein Info
Gene SymbolP2RY12
Full NamePurinergic Receptor P2Y12
AliasesP2RY12PROTEIN
Chromosome3q25.1-q25.2
Protein TypeGpcr
Target ClassGpcr
FunctionP2RY12 is a Gi/o protein-coupled receptor for ADP that plays a critical role in microglial surveillance and neuroimmune responses in the brain.
Mechanism of ActionP2Y12 receptor antagonists blocking ADP-mediated signaling
Subcellular Localization</b></td><td>Plasma Membrane, Microglial Processes</td></tr>
DruggabilityMedium (0.55)
Clinical StageApproved
PathwaysPI3K, MAPK
UniProt IDQ9H244
NCBI Gene ID29128
Ensembl IDENSG00000170017
GeneCardsP2RY12
Human Protein AtlasP2RY12
Associated DiseasesAD, ALS, AMI, ARM, Aging
Known Drugs/Compoundsstatins, rapamycin
InteractionsAPOA1, ULK1, ATG5, EIF4EBP1, LC3, MTOR
SciDEX TargetView Target Profile (8 clinical trials)
SciDEX HypothesesMicroglial Purinergic Reprogramming
Purinergic P2Y12 Inverse Agonist Therapy
KG Connections555 knowledge graph edges
DatabasesGeneCardsHPASTRING

Knowledge Graph

Related Hypotheses (20)

Microglial Purinergic Reprogramming
Score: 0.48
Purinergic P2Y12 Inverse Agonist Therapy
Score: 0.48
TREM2-Dependent Microglial Senescence Transition
Score: 0.69
Circadian Glymphatic Entrainment via Targeted Orexin Recepto
Score: 0.62
APOE-Dependent Autophagy Restoration
Score: 0.61

Related Analyses (14)

Neuroinflammation and microglial priming in early Alzheimer'
neurodegeneration · archived
What determines P2RY12 receptor expression/activity specific
neurodegeneration · failed
How does P2RY12-mediated VSMC dysfunction contribute to cere
neurodegeneration · failed
TDP-43 phase separation therapeutics for ALS-FTD
neurodegeneration · archived
Blood-brain barrier transport mechanisms for antibody therap
neurodegeneration · archived

Related Experiments (6)

s:** - GPR32 knockout in microglia should worsen neuroinflam
falsification · proposed · Score: 0.40
Proposed experiment from debate on Synaptic pruning by micro
falsification · proposed · Score: 0.40
FTD Microglia Role: Protective vs Destructive Mechanism Stud
validation · proposed · Score: 0.40
Purinergic Signaling Dysfunction Validation in Parkinson's D
clinical · proposed · Score: 0.40
Microglial TREM2 Agonist In Vivo Efficacy
validation · proposed · Score: 0.40

See Also (1)

Neurodegeneration
disease · KG edge: implicated_in