gene 2,157 words KG: EPHB4 2026-03-27
kind:genesection:genesstate:publishedevidence:strong
Contents

EPHB4 Gene

🧬 Gene Info
Gene SymbolEPHB4
AliasesEph Receptor B4
Chromosome5q22.1
Protein TypeKinase
Target ClassKinase
FunctionSmall molecule inhibitor of receptor tyrosine kinase activity
Mechanism of ActionSmall molecule inhibitor of receptor tyrosine kinase activity
Primary Expressionthe ventricular zone and cortical plate, coinciding with periods of active neurogenesis and neuronal migration
DruggabilityLow (0.43)
Clinical StageApproved
PathwaysEphrin-EphB receptor signaling
UniProt IDP54760
NCBI Gene ID2050
Ensembl IDENSG00000196411
OMIM600010
GeneCardsEPHB4
Human Protein AtlasEPHB4
Associated DiseasesAD, ALI, ALS, Cancer, Cardiac
Known Drugs/CompoundsIcariin
InteractionsSRC, RHOA, AKT, TP53, EFNB1, USH2A
SciDEX TargetView Target Profile (7 clinical trials)
SciDEX HypothesesEphrin-B2/EphB4 Axis Manipulation
KG Connections188 knowledge graph edges
DatabasesGeneCardsHPASTRING

Knowledge Graph

Related Hypotheses (19)

Ephrin-B2/EphB4 Axis Manipulation
Score: 0.40
Selective Acid Sphingomyelinase Modulation Therapy
Score: 0.68
CYP46A1 Overexpression Gene Therapy
Score: 0.66
APOE-Dependent Autophagy Restoration
Score: 0.63
SASP-Driven Aquaporin-4 Dysregulation
Score: 0.59

Related Analyses (6)

Neuroinflammation resolution mechanisms and pro-resolving me
neurodegeneration · archived
Lipid raft composition changes in synaptic neurodegeneration
neurodegeneration · completed
Synaptic pruning by microglia in early AD
neurodegeneration · archived
4R-tau strain-specific spreading patterns in PSP vs CBD
neurodegeneration · archived
Circuit-level neural dynamics in neurodegeneration
neuroscience · archived

Related Experiments (5)

Spatial transcriptomic analysis of multistage ESCC developme
exploratory · proposed · Score: 0.85
Functional analysis of EFNB1-EPHB4 interaction in EMT
exploratory · proposed · Score: 0.80
Analysis of TP53-TP63/ΔNP63-EFNB1-EPHB4 axis in cancer progr
exploratory · proposed · Score: 0.75
s:** - Test tau spreading in AQP4 knockout vs wild-type mice
falsification · proposed · Score: 0.40
s:** - Compare tau strain spreading in EXT1/EXT2 conditional
falsification · proposed · Score: 0.40

See Also (9)

Packard Center for ALS Research
institution · KG edge: activates
Accelerating Medicines Partnership for Alzheimer's Dise
institution · KG edge: implicated_in
APOE contributes to Alzheimer's disease by regulating b
hypothesis · KG edge: associated_with
CERS2 — Ceramide Synthase 2 (Lass2)
gene · KG edge: co_discussed
C1QA Gene
gene · KG edge: co_discussed

Knowledge Graph (12 edges)

EPHB4 interacts_with RASA1
EPHB4 associated_with VEIN OF GALEN MALFORMATION
EPHB4 associated_with TP53
EPHB4 mediates RASA1
EPHB4 causes RASA1
EPHB4 expressed_in RHOA
EPHB4 associated_with CANCER
EPHB4 associated_with neurodegeneration
EPHB4 co_discussed SMPD1
EPHB4 co_discussed C1QA