gene 711 words KG: GJA1 2026-03-22
kind:genesection:genesstate:published
Contents

GJA1

🧬 Gene Info
Gene SymbolGJA1
Full NameGap Junction Protein Alpha 1
Chromosome6q22.31
Protein FamilyConnexin family (21 members in humans)
Protein TypeChannel
Target ClassIon Channel
FunctionConnexin-43 forms gap junction channels enabling direct cell-to-cell transfer of ions (Ca²+, K+), small metabolites (ATP, glucose, glutamate), and signaling molecules.
Mechanism of ActionSmall molecule modulator of gap junction channel activity
DruggabilityLow (0.36)
Clinical StagePhase II
Molecular Weight43 kDa
PathwaysAutophagy, Blood-brain barrier function, Nf-Κb, Oxidative Stress, Proteasome
UniProt IDP17302
NCBI Gene ID2697
Ensembl IDENSG00000152661
OMIM121014
GeneCardsGJA1
Human Protein AtlasGJA1
Associated DiseasesAlzheimer, Alzheimer'S Disease, Amyloidosis, Cardiac, Chronic Non-Healing Wounds
Known Drugs/CompoundsBleomycin, Gap26
InteractionsTERT, PROGRANULIN, AQP4, GRN, APOE, SLC1A2
SciDEX TargetView Target Profile (2 clinical trials)
SciDEX HypothesesAstroglial Gap Junction Coordination via Connexin-
Astrocytic Connexin-43 Upregulation Enhances Neuro
CX43 hemichannel engineering enables size-selectiv
KG Connections702 knowledge graph edges
DatabasesGeneCardsHPASTRING

Knowledge Graph

Related Hypotheses (30)

Astroglial Gap Junction Coordination via Connexin-43 Phospho
Score: 0.50
CX43 hemichannel engineering enables size-selective mitochon
Score: 0.41
Astrocytic Connexin-43 Upregulation Enhances Neuroprotective
Score: 0.45
Context-Dependent Cx43 Modulation Based on Disease Stage
Score: 0.58
TNF-α/IL-1β-Cx43 Hemichannel Axis as Upstream Link Between S
Score: 0.55

Related Analyses (10)

Mitochondrial transfer between neurons and glia
neurodegeneration · archived
Mitochondrial transfer between astrocytes and neurons
neurodegeneration · archived
Perivascular spaces and glymphatic clearance failure in AD
neurodegeneration · archived
Microglia-astrocyte crosstalk amplification loops in neurode
neurodegeneration · archived
Sleep disruption as cause and consequence of neurodegenerati
neurodegeneration · archived

Related Experiments (10)

Cx43 knockdown effects on mitochondrial transfer
exploratory · proposed · Score: 0.90
Confocal imaging of MSC-chondrocyte interactions during mito
exploratory · proposed · Score: 0.85
Cx43 and GJA1-20k overexpression effects on mitochondrial tr
exploratory · proposed · Score: 0.95
Astrocyte Ferritin Iron Metabolism Dysfunction in Parkinson'
clinical · proposed · Score: 0.40
Gap Junction Dysfunction Validation in Parkinson's Disease
clinical · proposed · Score: 0.40

See Also (7)

Aging vs Neurodegeneration: Mechanistic Comparison Matr
mechanism · KG edge: biomarker_for
Alzheimer Indonesia
institution · KG edge: biomarker_for
APOE contributes to Alzheimer's disease by regulating b
hypothesis · KG edge: activates
AQP4 (Aquaporin-4 Gene)
gene · KG edge: activates
AQP1 Gene
gene · KG edge: co_discussed

Knowledge Graph (12 edges)

GJA1 associated_with neurodegeneration
GJA1 co_discussed HCRTR2
GJA1 co_discussed LOXL1-4
GJA1 co_discussed HCRTR1
GJA1 co_discussed AQP4
GJA1 co_discussed LOX
GJA1 co_discussed SDC1
GJA1 co_discussed PDGFRB
GJA1 co_discussed RAB27A
GJA1 co_discussed GAP43